N
H
HO
H
2
N
N
H
HO
H
2
N
N
H
HO
H
2
N
Spiroperidol
Spiperone
Iodocyanopindolol
(5-HT 1B)
Rauwolscine
(5-HT 1D)
8-OH-DPAT
8-OH-DPAT
LSD
5-CT
GIRK
Ca
2+
Ca
2+
5-HT1A
5-HT1B-1F
5-HT5
5-HT4
5-HT6
5-HT7
cAMP
PKA
Raf
PKC
MEK
MAPK
ERK1/2
AC
ATP
p90 RSK2
CREB
CRE
PIP
2
IP
3
DAG
BDNF
β-arr
γ
β
γ
β
γ
β
αi/0
αs
LSD
Mesulergine
Serotonylation of Rab Proteins
5-HT2A
5-HT2B
5-HT2C
SERT
γ
PLCβ
PLCγ
PH
Src
PLA
2
PLD
Arachidonic Acid
Phosphatidylcholine
Phosphatidic Acid
RhoA-GEF
RhoA
γ
β
β
αq/11
α12/13
NF-κB
PI3K
Akt
PKA
ERK1/2
MAPK
MEK
Raf
Ras
5-HT Receptor Antagonists
Clozapine
Olanzapine
Ketanserin
5-HT Receptor Agonists
Prucalopride
WAY-100635
Eletriptan
Pan-MEK Inhibitors
Trametinib
U0126-EtOH
PD184352
Selective MEK Inhibitors
Selumetinib (MEK1)
BIX 02189 (MEK5)
PKA Inhibitors
A-674563
H 89
AT13148
Pan-Akt Inhibitors
MK-2206
Perifosine
GSK690693
Selective Akt Inhibitors
A-674563 (Akt1)
CCT128930 (Akt2)
Rho Family Inhibitors
Zoledronic Acid
NSC 23766
EHop-016
ZCL278
PKA Inhibitors
A-674563
H 89
AT13148
ERK Inhibitors
SCH772984
XMD8-92
FR 180204
GDC-0994
cAMP Activator
Forskolin
P
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GIRK
Mesulergine
SERT
Serotonylation of Rab Proteins
Arachidonic Acid
Phosphatidylcholine
Phosphatidic Acid
8-OH-DPAT
Spiroperidol
Spiperone
Iodocyanopindolol
(5-HT 1B)
Rauwolscine
(5-HT 1D)
8-OH-DPAT
LSD
5-CT
LSD
Ca
Ca
2+
2+
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2
2
3
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Notes:
1:Clickable
2:Unclickable