13
12
10
11
2
3
6
8
7
4
5
1
9
9
F
usion
CD4
Co-receptor (CCR5 or CXCR4)
Host Cell
Budding
Matu
r
ation
ALIX,
ESC
R
T
-I,
ESC
R
T
-III
Attachment
Env
HIV-1
Uncoating
R
e
v
erse
T
r
anscription
Nuclear
Export
Nuclear
Import
Tat
Rev
Vpu
Vif
RNA
P
ol II
P-TEFb
T
r
anslation
T
r
anscription
Release
AAA
AAA
AAA
AAA
AAA
AAA
AAA
AAA
AAA
5’
L
TR
3’
L
TR
Integ
r
ation
LEDGF
Accessory Vi
r
al
P
r
oteins
Assembly
Pre-integration
Complex
Gag
Gag
P
ol
T
r
anslation
Gag
Gag
P
ol
HIV Protease Inhibitors
Pepstatin A
Nelfinavir
Ritonavir
Lopinavir
Pan-CXCR Antagonist
Reparixin
Selective-CXCR Antagonists
Plerixafor (CXCR4)
SB225002 (CXCR2)
WZ811 (CXCR4)
CCR Antagonist
Maraviroc (CCR5)
CCR Agonist
ZK756326 (CCR8)
Integrase Inhibitors
Raltegravir
Dolutegravir
Elvitegravir
Cabotegravir
Bictegravir
Reverse Transcriptase
Inhibitors
Lamivudine
Emtricitabine
Tenofovir
Zidovudine
Efavirenz
CRM1 Inhibitors
Selinexor
Eltanexor
KPT-185
Verdinexor
P
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Notes:
1:Clickable
2:Unclickable